PAT-IN-2
PAT-IN-2 is a protein acyl transferases (PAT) inhibitor. PAT-IN-2 competitively inhibits Erf2 autopalmitoylation (WO2017011518A1; compound 25).
For research use only. We do not sell to patients.
- CAS No.: 2066572-01-6
- Formula: C42H56F6N4O
- Molecular Weight:746.91
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
PAT-IN-2 (compound 25) completely inhibits growth of RJY1941 (control) at 20 μΜ, but has no detectable effect at lower concentrations. PAT-IN-2 inhibits the growth of RJY1942 (palmitoylation sensitive) at 5 μΜ[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS No. 2066572-01-6
-
Molecular Weight 746.91
-
Formula C42H56F6N4O
-
SMILES
CC(C1=CC=C(C=C1)CC(C)C)CN(CCN(C2)CCCC[C@@H]3N(CCNC3)CCC4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)[C@H]2CC5=CC=C(C=C5)O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)