1. Cell Cycle/DNA Damage
  2. PERK
  3. PERK-IN-4

PERK-IN-4 

Cat. No.: HY-137813
Handling Instructions

PERK-IN-4 is a potent and selective PERK (protein kinase R (PKR)-like endoplasmic reticulum kinase) inhibitor with an IC 50 of 0.3 nM. PERK is activated in response to a variety of endoplasmic reticulum stresses implicated in numerous disease states.

For research use only. We do not sell to patients.

PERK-IN-4 Chemical Structure

PERK-IN-4 Chemical Structure

CAS No. : 1337531-89-1

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Description

PERK-IN-4 is a potent and selective PERK (protein kinase R (PKR)-like endoplasmic reticulum kinase) inhibitor with an IC 50 of 0.3 nM. PERK is activated in response to a variety of endoplasmic reticulum stresses implicated in numerous disease states[1].

IC50 & Target

IC50: 0.3 nM (PERK)[1]

Molecular Weight

469.43

Formula

C₂₄H₁₉F₄N₅O

CAS No.
Shipping

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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PERK-IN-4
Cat. No.:
HY-137813
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