1. Others
  2. Others
  3. (Rac)-BMS-816336

(Rac)-BMS-816336 

Cat. No.: HY-101930A
Handling Instructions

(Rac)-BMS-816336 (Compound 6n)is a racemate of BMS-816336. (Rac)-BMS-816336 is a potent inhibitor of human and mouse 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) enzyme with IC50s of 10 nM and 68 nM, respectively. (Rac)-BMS-816336 has good metabolic stability.

For research use only. We do not sell to patients.

(Rac)-BMS-816336 Chemical Structure

(Rac)-BMS-816336 Chemical Structure

Size Price Stock
10 mM * 1 mL in DMSO USD 265 Ask For Quote & Lead Time
5 mg USD 350 Ask For Quote & Lead Time
10 mg USD 550 Ask For Quote & Lead Time
50 mg USD 1650 Ask For Quote & Lead Time
100 mg USD 2650 Ask For Quote & Lead Time

* Please select Quantity before adding items.

Other In-stock Forms of (Rac)-BMS-816336:

Other Forms of (Rac)-BMS-816336:

Top Publications Citing Use of Products
  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

(Rac)-BMS-816336 (Compound 6n)is a racemate of BMS-816336. (Rac)-BMS-816336 is a potent inhibitor of human and mouse 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) enzyme with IC50s of 10 nM and 68 nM, respectively. (Rac)-BMS-816336 has good metabolic stability[1].

IC50 & Target

IC50: 10 nM (Human 11β-HSD1) and 68 nM (Mouse 11β-HSD1)[1]

In Vivo

(Rac)-BMS-816336 (compound 6n) has good metabolic stability, and the remaining rates in human, mouse and rats of 88%,82% and 72%, respectively[1].

Molecular Weight

341.44

Formula

C₂₁H₂₇NO₃

SMILES

OC1[[email protected]]2C[[email protected]@H]3[[email protected]@](C4=CC=CC=C4)(CC(N5CC(O)C5)=O)[[email protected]@H](CC1C3)C2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • No file chosen (Maximum size is: 1024 Kb)
  • If you have published this work, please enter the PubMed ID.
  • Your name will appear on the site.
  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

(Rac)-BMS-816336Others11β-HSD1BMS-816336racematemetabolicstabilityInhibitorinhibitorinhibit

Your Recently Viewed Products:

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country or Region *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product name:
(Rac)-BMS-816336
Cat. No.:
HY-101930A
Quantity:
MCE Japan Authorized Agent: