1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. GABA Receptor
  3. Radequinil

Radequinil (Synonyms: AC-3933)

Cat. No.: HY-106025
Handling Instructions

Radequinil (AC-3933) is a benzodiazepine receptor (BzR) partial inverse agonist. AC-3933 binds to GABA(-) and GABA(+) ligand with Kis of 5.15 and 6.11 nM, respectively.

For research use only. We do not sell to patients.

Radequinil Chemical Structure

Radequinil Chemical Structure

CAS No. : 219846-31-8

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Description

Radequinil (AC-3933) is a benzodiazepine receptor (BzR) partial inverse agonist. AC-3933 binds to GABA(-) and GABA(+) ligand with Kis of 5.15 and 6.11 nM, respectively[1].

IC50 & Target

Ki: 5.15±0.39 nM (GABA(-) ligand), 6.11±0.26 nM (GABA(+) ligand)[1]

Clinical Trial
Molecular Weight

334.33

Formula

C₁₈H₁₄N₄O₃

CAS No.

219846-31-8

SMILES

O=C1NC2=CC=NC(C3=CC(OC)=CC=C3)=C2C=C1C4=NOC(C)=N4

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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