S1427
S1427 is a tranylcypromine-derived LSD1 inhibitor with the IC50 of 390 nM and Ki of 80 nM. S1427 exhibits desirable hERG channel inhibition and microsomal stability profiles. Inhibition of LSD1 partially reduces the proliferation of cancer cells.
For research use only. We do not sell to patients.
- CAS No.: 2447061-40-5
- Formula: C25H29F3N4O2
- Molecular Weight:474.52
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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KDM1/LSD1 |
Chemical Information
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CAS No. 2447061-40-5
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Molecular Weight 474.52
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Formula C25H29F3N4O2
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SMILES
O=C(N1CCC2(CC1)CCNC2)CN[C@H]3C[C@@H]3C4=C(C(F)=CC(F)=C4)OCC5=CC=CN=C5F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)