Setastine
Based on 1 Customer Validation
Setastine (EGIS-2062 (free acid); EGYT-2062 (free acid) is an orally effective, non-sedative and long acting anti-allergic agent. Setastine possesses potent histamine Hi-receptor blocking properties and can be used for allergies and rhinitis research[1]<.
For research use only. We do not sell to patients.
- Purity: 99.21%
- CAS No.: 64294-95-7
- Formula: C22H28ClNO
- Molecular Weight:357.92
-
Storage:Pure form -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
-
Biological Activity
-
Chemical Information
-
Solvent & Solubility
- Purity & Documentation
- References
-
Help & FAQs
-
GPCR/G Protein Compound Library
HY-L006
-
Immunology/Inflammation Compound Library
HY-L007
-
Neuronal Signaling Compound Library
HY-L013
-
Neurotransmitter Receptor Compound Library
HY-L062
-
Anti-Parkinson's Disease Compound Library
HY-L085
-
Neurodegenerative Disease-related Compound Library
HY-L086
-
Anti-Obesity Compound Library
HY-L087
-
Protein-protein Interaction Inhibitor Library
HY-L109
-
Coagulation and Anti-coagulation Compound Library
HY-L136
-
Membrane Protein-targeted Compound Library
HY-L149
-
Membrane Receptor-targeted Compound Library
HY-L150
-
Bioactive Compound Library Max
HY-L181
-
MCE Bioactive Compound Library
HY-L001V
-
Bioactive Compound Library
HY-L001
-
High-Throughput Bioactive Compound Library
HY-L205
-
Lactylation Compound Library
HY-L249
All Histamine Receptor Isoforms
More
Biological Activity
IC50:Histamine Hi-receptor[1]
Chemical Information
-
CAS No. 64294-95-7
-
Appearance Liquid
-
Molecular Weight 357.92
-
Formula C22H28ClNO
-
Color Colorless to light yellow
-
SMILES
CC(C1=CC=C(C=C1)Cl)(OCCN2CCCCCC2)C3=CC=CC=C3
-
Synonyms
EGIS-2062 free acid; EGYT-2062 free acid
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Pure form -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : ≥ 125 mg/mL (349.24 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
-
Data Sheet (271 KB)
-
SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Portuguese - PT (252 KB)
-
Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.7939 mL | 13.9696 mL | 27.9392 mL | 69.8480 mL |
| 5 mM | 0.5588 mL | 2.7939 mL | 5.5878 mL | 13.9696 mL | |
| 10 mM | 0.2794 mL | 1.3970 mL | 2.7939 mL | 6.9848 mL | |
| 15 mM | 0.1863 mL | 0.9313 mL | 1.8626 mL | 4.6565 mL | |
| 20 mM | 0.1397 mL | 0.6985 mL | 1.3970 mL | 3.4924 mL | |
| 25 mM | 0.1118 mL | 0.5588 mL | 1.1176 mL | 2.7939 mL | |
| 30 mM | 0.0931 mL | 0.4657 mL | 0.9313 mL | 2.3283 mL | |
| 40 mM | 0.0698 mL | 0.3492 mL | 0.6985 mL | 1.7462 mL | |
| 50 mM | 0.0559 mL | 0.2794 mL | 0.5588 mL | 1.3970 mL | |
| 60 mM | 0.0466 mL | 0.2328 mL | 0.4657 mL | 1.1641 mL | |
| 80 mM | 0.0349 mL | 0.1746 mL | 0.3492 mL | 0.8731 mL | |
| 100 mM | 0.0279 mL | 0.1397 mL | 0.2794 mL | 0.6985 mL |
Powered by Bioz