FSLLRY-NH2
Based on 6 publication(s) in Google Scholar
FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.
For research use only. We do not sell to patients.
- Purity: 99.89%
- CAS No.: 245329-02-6
- Formula: C39H60N10O8
- Molecular Weight:796.96
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Storage:
Sealed storage, away from moisture and light.
Powder -80°C, 2 years , -20°C, 1 year* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
Publications Citing Use of MedChemExpress (MCE) FSLLRY-NH2
More
Biological Activity
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PAR2 |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 245329-02-6
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Appearance Solid
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Molecular Weight 796.96
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Formula C39H60N10O8
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Color White to off-white
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Sequence
Phe-Ser-Leu-Leu-Arg-Tyr-NH2
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Sequence Shortening
FSLLRY-NH2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Sealed storage, away from moisture and light
Powder -80°C 2 years -20°C 1 year * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
Publications (6)
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Journal Impact Factor
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Most Recent
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J Immunother Cancer
Unveiling the mechanisms of CEBPD-orchestrated TAM polarization through RGS2/PAR2 pathway and its impact on ICB efficacy in clear cell renal cell carcinoma. [Abstract]2025 Jul 13;13(7):e010898. PMID: 40659446 -
Brain Behav Immun
2024 Jun 12:120:403-412. PMID: 38871062 -
Biomolecules
PAR2 Participates in the Development of Cough Hypersensitivity in Guinea Pigs by Regulating TRPA1 Through PKC. [Abstract]2025 Feb 1;15(2):208. PMID: 40001511 -
Cell Signal
Angiotensin II depends on hippo/YAP signaling to reprogram angiogenesis and promote liver fibrosis. [Abstract]2024 Nov:123:111355. PMID: 39173854 -
BMC Musculoskelet Disord
Knockdown of PAR2 alleviates cancer-induced bone pain by inhibiting the activation of astrocytes and the ERK pathway. [Abstract]2022 May 30;23(1):514. PMID: 35637468 -
Solvent & Solubility
DMSO : 100 mg/mL (125.48 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (272 KB)
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SDS (394 KB)
- English - EN (394 KB)
- Français - FR (394 KB)
- Deutsch - DE (394 KB)
- Norwegian - NO (394 KB)
- Español - ES (394 KB)
- Swedish - SV (394 KB)
- Italian - IT (394 KB)
- Korean - KR (394 KB)
- Portuguese - PT (394 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.2548 mL | 6.2738 mL | 12.5477 mL | 31.3692 mL |
| 5 mM | 0.2510 mL | 1.2548 mL | 2.5095 mL | 6.2738 mL | |
| 10 mM | 0.1255 mL | 0.6274 mL | 1.2548 mL | 3.1369 mL | |
| 15 mM | 0.0837 mL | 0.4183 mL | 0.8365 mL | 2.0913 mL | |
| 20 mM | 0.0627 mL | 0.3137 mL | 0.6274 mL | 1.5685 mL | |
| 25 mM | 0.0502 mL | 0.2510 mL | 0.5019 mL | 1.2548 mL | |
| 30 mM | 0.0418 mL | 0.2091 mL | 0.4183 mL | 1.0456 mL | |
| 40 mM | 0.0314 mL | 0.1568 mL | 0.3137 mL | 0.7842 mL | |
| 50 mM | 0.0251 mL | 0.1255 mL | 0.2510 mL | 0.6274 mL | |
| 60 mM | 0.0209 mL | 0.1046 mL | 0.2091 mL | 0.5228 mL | |
| 80 mM | 0.0157 mL | 0.0784 mL | 0.1568 mL | 0.3921 mL | |
| 100 mM | 0.0125 mL | 0.0627 mL | 0.1255 mL | 0.3137 mL |