TC OT 39
Based on 1 Customer Validation
TC OT 39 is a synthetic oxytocin analog, as well as a selective agonist of oxytocin receptor (OXTR, EC50=180 nM). TC OT 39 is also an Avprla vasopressin receptor antagonist with an Ki value of 330 nM. TC OT 39 exhibits sedative effects in mouse models.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- Purity : 97.7%
- CAS No.: 479232-57-0
- 화학식: C32H40N8O2S
- 분자량:600.78
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보관:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- 순도&문서
- References
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Help & FAQs
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AtosibanOxytocin/Vasopressin Receptor Antagonist -
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WAY-267464Oxytocin Receptor (OTR) Agonist -
HY-17573
CarbetocinOxytocin Receptor Agonist -
HY-15015
OT-R antagonist 1Oxytocin Receptor Antagonist -
HY-108677R
L-368,899 hydrochloride (Standard)Reference Standard -
![[Asp5]-Oxytocin](https://file.medchemexpress.com/product_pic/hy-p3217.gif)
HY-P3217
[Asp5]-OxytocinNeurohypophyseal Hormone Analogue -
HY-15023
CligosibanOxytocin Receptor Antagonist -
HY-17572R
Atosiban (Standard)Oxytocin/Vasopressin Receptor Antagonist
All Vasopressin Receptor Isoforms
More
Biological Activity
제품 설명
IC50 & Target
[1]|
Avprla vasopressin receptor 300 nM (Ki) |
Oxytocin Receptor 180 nM (EC50) |
Cellular Effect
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Cell Line
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Type | Value | Description | References |
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| CHO | EC50 |
33 nM
Compound: 1
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Activity at human oxytocin receptor expressed in CHO cells by NFAT-luciferase gene reporter assay
Activity at human oxytocin receptor expressed in CHO cells by NFAT-luciferase gene reporter assay
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[PMID: 20104850] |
| CHO | EC50 |
850 nM
Compound: 1
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Activity at human vasopressin V2 receptor expressed in CHO cells by NFAT-luciferase gene reporter assay
Activity at human vasopressin V2 receptor expressed in CHO cells by NFAT-luciferase gene reporter assay
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[PMID: 20104850] |
In Vivo
Marble burying is based on the natural instinct of rodents to bury objects, commonly used in preclinical research to assess anxiety-like behavior in rodents[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 479232-57-0
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Appearance Solid
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분자량 600.78
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화학식 C32H40N8O2S
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Color White to off-white
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SMILES
O=C(N1[C@H](C(N2CCN(C)CCC2)=S)CCC1)NCC3=CC=C(C(N4CC5=C(N(C)N=C5)NC6=CC=CC=C46)=O)C=C3C
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
순도&문서
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Data Sheet (268 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
TC OT 39 Related Classifications
HY-108678 Related Classifications
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