1. GPCR/G Protein
    Neuronal Signaling
  2. Cannabinoid Receptor
  3. Tedalinab

Tedalinab (Synonyms: GRC-10693)

Cat. No.: HY-14900
Handling Instructions

Tedalinab (GRC-10693) is a potent, orally active, and selective cannabinoid receptor 2 (CB2) agonist. Tedalinab has >4700-fold functional selectivity for CB2 over CB1. Tedalinab has potential for neuropathic pain and osteoarthritis treatment.

For research use only. We do not sell to patients.

Tedalinab Chemical Structure

Tedalinab Chemical Structure

CAS No. : 916591-01-0

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Description

Tedalinab (GRC-10693) is a potent, orally active, and selective cannabinoid receptor 2 (CB2) agonist. Tedalinab has >4700-fold functional selectivity for CB2 over CB1. Tedalinab has potential for neuropathic pain and osteoarthritis treatment[1].

IC50 & Target[1]

CB2

 

Molecular Weight

345.39

Formula

C₁₉H₂₁F₂N₃O

CAS No.

916591-01-0

SMILES

O=C(C1=NN(C2=CC=C(F)C=C2F)C3=C1[[email protected]@]4([H])CC[[email protected]]3([H])C4)NC(C)(C)C

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

TedalinabGRC-10693GRC10693GRC 10693Cannabinoid ReceptorneuropathicpainosteoarthritisselectiveoralbioavailabilityInhibitorinhibitorinhibit

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