1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. iGluR
  3. UBP 302

UBP 302 

Cat. No.: HY-107604 Purity: >99.0%
Handling Instructions

UBP 302 is a potent and selective GLUK5-subunit containing kainate receptor antagonist (apparent Kd=402 nM), and displays very little affinity on GluK2 (GluR6) kainate receptors. Anxiolytic effects.

For research use only. We do not sell to patients.

UBP 302 Chemical Structure

UBP 302 Chemical Structure

CAS No. : 745055-91-8

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 477 In-stock
Estimated Time of Arrival: December 31
5 mg USD 650 In-stock
Estimated Time of Arrival: December 31
10 mg USD 1100 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

UBP 302 is a potent and selective GLUK5-subunit containing kainate receptor antagonist (apparent Kd=402 nM), and displays very little affinity on GluK2 (GluR6) kainate receptors. Anxiolytic effects[1][2][3].

IC50 & Target

apparent Kd: 402 nM (GLUK5)[2]
IC50: 106 μM (AMPA receptors)[2]

Molecular Weight

333.30

Formula

C₁₅H₁₅N₃O₆

CAS No.

745055-91-8

SMILES

O=C(N(C=CC1=O)C[[email protected]](N)C(O)=O)N1CC2=C(C=CC=C2)C(O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References

Purity: >99.0%

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Keywords:

UBP 302UBP302UBP-302iGluRIonotropic glutamate receptorsInhibitorinhibitorinhibit

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UBP 302
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HY-107604
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