VUF14480
VUF14480 is a partial agonist of histamine H4 (hH4) receptor-mediated G protein signalling and β-arrestin2 recruitment. VUF14480 binds covalently to hH4 receptor (pKi: 6.3 for hH4-WT receptor). VUF14480 partially induces hH4 receptor-mediated G protein activation and β-arrestin2 recruitment. VUF14480 can be used in the research of inflammatory diseases.
For research use only. We do not sell to patients.
- CAS No.: 1605304-31-1
- Formula: C17H20N4
- Molecular Weight:280.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Histamine Receptor Isoforms
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Biological Activity
pKi: 6.3 for hH4-WT receptor[1]
Chemical Information
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CAS No. 1605304-31-1
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Molecular Weight 280.38
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Formula C17H20N4
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SMILES
N=1C(=NC(=CC1C=2C=CC=CC2)N3CCN(C)CC3)C=C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
VUF14480 Related Classifications
HY-165453 Related Classifications
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