1. Neuronal Signaling
  2. CaMK

CaMKII-IN-1 

Cat. No.: HY-18271 Purity: 98.09%
Handling Instructions

CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM; significantly high selectivity against CaMKIV, MLCK, p38a, Akt1, and PKC.

For research use only. We do not sell to patients.

CaMKII-IN-1 Chemical Structure

CaMKII-IN-1 Chemical Structure

CAS No. : 1208123-85-6

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 506 In-stock
Estimated Time of Arrival: December 31
5 mg USD 420 In-stock
Estimated Time of Arrival: December 31
10 mg USD 600 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1800 In-stock
Estimated Time of Arrival: December 31
100 mg USD 2520 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM; significantly high selectivity against CaMKIV, MLCK, p38a, Akt1, and PKC. IC50 value: 63 nM Target: CaMKII

Solvent & Solubility
In Vitro: 

DMSO : ≥ 54 mg/mL (98.52 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.8245 mL 9.1224 mL 18.2448 mL
5 mM 0.3649 mL 1.8245 mL 3.6490 mL
10 mM 0.1824 mL 0.9122 mL 1.8245 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

548.10

Formula

C₂₉H₃₀ClN₅O₂S

CAS No.

1208123-85-6

SMILES

O=S(C1=CC=CC(Cl)=C1C)(NC2=C(CN(CC3=CC=CC=C3)CC4)C4=NC(NCCC5=CC=CC=C5)=N2)=O

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
CaMKII-IN-1
Cat. No.:
HY-18271
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CaMKII-IN-1

Cat. No.: HY-18271