1. Metabolic Enzyme/Protease
  2. Acyltransferase
  3. FR-190809

FR-190809 

Cat. No.: HY-122078
Handling Instructions

FR-190809 is a potent, nonadrenotoxic, orally efficacious acyl-CoA:cholesterol O-acyltransferase (ACAT) inhibitor, with an IC50 of 45 nM.

For research use only. We do not sell to patients.

FR-190809 Chemical Structure

FR-190809 Chemical Structure

CAS No. : 215589-63-2

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Description

FR-190809 is a potent, nonadrenotoxic, orally efficacious acyl-CoA:cholesterol O-acyltransferase (ACAT) inhibitor, with an IC50 of 45 nM[1].

IC50 & Target

IC50: (ACAT)[1]

In Vitro

FR-190809 inhibits foam cell formation with an IC50 of 215 nM[1].

Molecular Weight

603.73

Formula

C₂₉H₃₄FN₃O₆S₂

CAS No.

215589-63-2

SMILES

O=C(NC1=C(S(=O)(C)=O)C=C(C)N=C1S(=O)(C)=O)N(C2CCCCCC2)CC3=CC=C(OC4=CC=C(F)C=C4)C=C3

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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FR-190809
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HY-122078
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