1. GPCR/G Protein
  2. Adenosine Receptor
  3. MRS1177

MRS1177 

Cat. No.: HY-120090
Handling Instructions

MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM.

For research use only. We do not sell to patients.

MRS1177 Chemical Structure

MRS1177 Chemical Structure

CAS No. : 183721-13-3

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Description

MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM.

IC50 & Target

Ki: 0.3 nM (hA3AR)[1][2].

In Vitro

MRS1177 (compound 2b) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist[1]. The Ki value of MRS1177 (compound 55) with hA3AR is 0.3 nM[2].

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

389.79

Formula

C₂₀H₁₂ClN₅O₂

CAS No.

183721-13-3

SMILES

O=C(C1=CC=CC=C1)NC2=NC3=C(C4=NC(C5=CC=CO5)=NN24)C=C(C=C3)Cl

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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Product Name:
MRS1177
Cat. No.:
HY-120090
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MRS1177

Cat. No.: HY-120090