1. GPCR/G Protein
  2. Adenosine Receptor

MRS1186 

Cat. No.: HY-118678
Handling Instructions

MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.

For research use only. We do not sell to patients.

MRS1186 Chemical Structure

MRS1186 Chemical Structure

CAS No. : 183721-03-1

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.

IC50 & Target

Ki: 7.66 nM (hA3AR)[1].

In Vitro

MRS1186 (compound 2d) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM[1].

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.9261 mL 14.6306 mL 29.2612 mL
5 mM 0.5852 mL 2.9261 mL 5.8522 mL
10 mM 0.2926 mL 1.4631 mL 2.9261 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

341.75

Formula

C₁₆H₁₂ClN₅O₂

CAS No.

183721-03-1

SMILES

CCC(NC1=NC2=C(C3=NC(C4=CC=CO4)=NN13)C=C(C=C2)Cl)=O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
MRS1186
Cat. No.:
HY-118678
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MRS1186

Cat. No.: HY-118678