1. Membrane Transporter/Ion Channel
  2. Sodium Channel
  3. PF-05241328

PF-05241328 

Cat. No.: HY-103623
Handling Instructions

PF-05241328 is a potent and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (Nav1.7), with an IC50 of 31 nM.

For research use only. We do not sell to patients.

PF-05241328 Chemical Structure

PF-05241328 Chemical Structure

CAS No. : 1387633-03-5

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Description

PF-05241328 is a potent and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (Nav1.7), with an IC50 of 31 nM.

IC50 & Target

IC50: 31 nM (Nav1.7)[1].

Clinical Trial
Molecular Weight

436.91

Formula

C₁₉H₂₁ClN₄O₄S

CAS No.

1387633-03-5

SMILES

O=C(C1=CC2=C(N(C3=CC(Cl)=C(OCC(C)C)N=C3)N=C2C)C=C1)NS(=O)(C)=O

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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PF-05241328
Cat. No.:
HY-103623
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