1. Metabolic Enzyme/Protease
  2. Dipeptidyl Peptidase

Retagliptin Phosphate (Synonyms: SP 2086)

Cat. No.: HY-112668 Purity: 99.69%
Handling Instructions

Retagliptin Phosphate is pharmaceutical composition of DPP-4 inhibitor for treating type-2 diabetes.

For research use only. We do not sell to patients.

Retagliptin Phosphate Chemical Structure

Retagliptin Phosphate Chemical Structure

CAS No. : 1256756-88-3

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 186 In-stock
Estimated Time of Arrival: December 31
5 mg USD 150 In-stock
Estimated Time of Arrival: December 31
10 mg USD 240 In-stock
Estimated Time of Arrival: December 31
50 mg USD 750 In-stock
Estimated Time of Arrival: December 31
100 mg USD 1200 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Retagliptin Phosphate is pharmaceutical composition of DPP-4 inhibitor for treating type-2 diabetes.

IC50 & Target

DPP-4[1].

Solvent & Solubility
In Vitro: 

DMSO : ≥ 150 mg/mL (266.73 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.7782 mL 8.8911 mL 17.7822 mL
5 mM 0.3556 mL 1.7782 mL 3.5564 mL
10 mM 0.1778 mL 0.8891 mL 1.7782 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (4.45 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (4.45 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (4.45 mM); Clear solution

References
Molecular Weight

562.36

Formula

C₁₉H₂₁F₆N₄O₇P

CAS No.

1256756-88-3

SMILES

O=C(C1=C2CN(C(C[[email protected]](N)CC3=CC(F)=C(F)C=C3F)=O)CCN2C(C(F)(F)F)=N1)OC.O=P(O)(O)O

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Purity: 99.69%

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Retagliptin Phosphate
Cat. No.:
HY-112668
Quantity:

Retagliptin Phosphate

Cat. No.: HY-112668