1. Metabolic Enzyme/Protease
  2. Phosphodiesterase (PDE)

Revizinone (Synonyms: R80122)

Cat. No.: HY-100615 Purity: 98.10%
Data Sheet SDS Handling Instructions

Revizinone is a novel selective phosphodiesterase (PDE) inhibitor with IC50 values on this enzyme to 0.036 microM.

For research use only. We do not sell to patients.
Revizinone Chemical Structure

Revizinone Chemical Structure

CAS No. : 133718-29-3

Size Price Stock Quantity
10 mM * 1 mL in DMSO $152 In-stock
1 mg $80 In-stock
5 mg $150 In-stock
10 mg $210 In-stock
50 mg $650 In-stock
100 mg $950 In-stock
200 mg   Get quote  
500 mg   Get quote  

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Other Forms of Revizinone:

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Description

Revizinone is a novel selective phosphodiesterase (PDE) inhibitor with IC50 values on this enzyme to 0.036 microM. target: phosphodiesterase (PDE)[3]; IC 50: 0.036 microM; [3] In vivo: The administration of Revizinone improved the haemodynamic profile with an increase in cardiac output, a decrease in systemic vascular resistance and a stable heart rate and mean arterial blood pressure. [1] With regard to reconstitution of contractility and cardiac function Revizinone (E-isomer) was 10 fold more potent than R 79595 and nearly 100 fold more potent than R 80123 (Z-isomer). [2] Revizinone significantly increased global LV function and systolic wall thickening in ischemic areas at doses greater than or equal to 0.16 mg/kg i.v. [4]

References
Molecular Weight

459.54

Formula

C₂₆H₂₉N₅O₃

CAS No.

133718-29-3

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

DMSO: ≥ 4.6 mg/mL

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

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Product Name:
Revizinone
Cat. No.:
HY-100615
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