Drug Derivative
Drug derivative
Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.
References:
- [1]. Vardanyan RS, et al. Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications. Future Med Chem. 2014 Mar;6(4):385-412.x
- [2]. Ghosh AK, et al. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry. J Med Chem. 2020 Mar 26;63(6):2751-2788.x
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Drug Derivative Inhibitors
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Drug Derivative Controls
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Drug Derivative Related Products (4062)
Related Products (4062)
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Cyclazodone
0 ImagesCat. No.: HY-116105CAS No.: 14461-91-7Cyclazodone is a neuroactive compound.
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Δ9-Tetrahydrocannabivarinic acid
0 ImagesCat. No.: HY-W775305CAS No.: 39986-26-0Synonyms: Δ9-THCVA-AΔ9-Tetrahydrocannabivarinic acid (THCVA) is a phytocannabinoid.
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ACEA1011
0 ImagesCat. No.: HY-116766CAS No.: 153504-72-4ACEA1011 is an active compound.
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Amogammadex
0 ImagesCat. No.: HY-159818CAS No.: 1309580-40-2Synonyms: Adamgammadex; Aom0498Amogammadex (Adamgammadex; Aom0498) is a modified γ-cyclodextrin (HY-W040040) derivative and neuromuscular blocking agent. Amogammadex forms inactive, tight inclusion complexes with free Rocuronium (HY-17033) and Vecuronium (HY-B0118A), and reverses the neuromuscular blockade induced by them in a concentration-dependent manner. Amogammadex can be used in research related to neuromuscular blockade reversal.
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Lachnone A
0 ImagesCat. No.: HY-126202CAS No.: 903892-99-9Lachnone A is a chromone derivative isolated from the filamentous fungus Lachnum sp. BCC 2424.
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Dulcoside C
0 ImagesCat. No.: HY-N18366CAS No.: 64432-09-3Dulcoside C is a rhamnose-containing steviol glycoside found in Stevia rebaudiana leaves.Dulcoside C exhibits significantly lower sweetness compared to Rebaudioside A (HY-N0466).
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N-Hydroxy MDMA hemioxalate
0 ImagesCat. No.: HY-172346Synonyms: N-OH MDMA hemioxalate; FLEA hemioxalateN-Hydroxy MDMA (N-OH MDMA) hemioxalate is an N-hydroxy analogue of 3,4-methylenedioxymethamphetamine (MDMA). N-Hydroxy MDMA hemioxalate can be rapidly metabolized to MDMA and MDA in rats, which are mainly excreted in urine, and can also be detected in hair.
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Bromothricin
0 ImagesCat. No.: HY-N16370Bromothricin is a brominated dervitaive of the macrolide antibiotic Chlorothricin (HY-125552). Bromothricin is a bacterial metabolite.
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9-Acetoxythymol
0 ImagesCat. No.: HY-N17549CAS No.: 216378-01-79-Acetoxythymol is a natural product that can be found in Thymus mongolicus?(Ronniger)?.
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Linalyl formate
0 ImagesCat. No.: HY-W791537CAS No.: 115-99-1Linalyl formate, an ester derivative of Linalool (HY-N0368), is one of the four main volatile substances in fresh blueberry juice
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Hyuganin A
0 ImagesCat. No.: HY-N17325CAS No.: 214778-42-4Hyuganin A is a natural product that can be found in Ilex rotunda?Thunb..
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Epimedonin K
0 ImagesCat. No.: HY-N9671CAS No.: 2222285-85-8Epimedonin K is a 2-phenoxychromone compound found in Epimedium brevicornum. Epimedonin K can be used for the research of cancer.
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Cucurbitacin V
0 ImagesCat. No.: HY-N13811CAS No.: 152340-37-9Cucurbitacin V is a natural triterpene.
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Musellarin C
0 ImagesCat. No.: HY-N16946CAS No.: 1392476-33-3Musellarin C is a natural phenolic compound.
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Souliene A
0 ImagesCat. No.: HY-N17066CAS No.: 1338332-32-3Souliene A is a natural sesquiterpene.
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JG-258
0 ImagesCat. No.: HY-148745CAS No.: 2241517-83-7JG-258 is an inactive negative control for Hsp70 inhibitors. JG-258 is an inactive structural analog of JG-98 (HY-117282), an allosteric inhibitor of heat shock protein 70 (Hsp70) with demonstrated anticancer activity. JG-258 can be used in cancer-related research.
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(+)-3β-Hydroxycarvotagenone
0 ImagesCat. No.: HY-N16604CAS No.: 120850-08-0(+)-3β-Hydroxycarvotagenone (Compound (4S,5R)-(−)-6a) is a α-phellandrene (HY-121615) derivative.
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Tanetin
0 ImagesCat. No.: HY-N13836CAS No.: 84019-17-0Tanetin is a natural flavonoid.
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Labda-12E,14-dien-16,15-olid-17-oic acid
0 ImagesCat. No.: HY-N17159CAS No.: 1855905-16-6Labda-12E,14-dien-16,15-olid-17-oic acid is a natural diterpene.
