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A2AAR antagonist 1 

Cat. No.: HY-151387
Handling Instructions

A2AAR antagonist 1 (compound 21a) is an A2AAR (adenosine A2A receptor) antagonist with a Ki value of 20 nM. A2AAR antagonist 1 shows high ligand efficiency, and it can be used for the research of neurodegenerative diseases.

For research use only. We do not sell to patients.

A2AAR antagonist 1 Chemical Structure

A2AAR antagonist 1 Chemical Structure

CAS No. : 1784491-64-0

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Description

A2AAR antagonist 1 (compound 21a) is an A2AAR (adenosine A2A receptor) antagonist with a Ki value of 20 nM. A2AAR antagonist 1 shows high ligand efficiency, and it can be used for the research of neurodegenerative diseases[1].

In Vitro

A2AAR antagonist 1 (0-10 μM; 1 h) shows a high affinity towards A2AAR with a Ki value of 20 nM[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

290.12

Formula

C12H8BrN3O

CAS No.
SMILES

NC1=NC(C2=CC=CO2)=C3C=C(Br)C=CC3=N1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
A2AAR antagonist 1
Cat. No.:
HY-151387
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