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Cat. No.: HY-179671

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A3AR antagonist 6

A3AR antagonist 6 (Compound 5p) is a selective A₃AR antagonist with a K_i of 6.8 nM. A3AR antagonist 6 can be used in tumor research.

For research use only. We do not sell to patients.

Formula: C₁₈H₂₀N₄O₅S
Molecular Weight:404.44

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (272 KB)

A3AR antagonist 6 Chemical Structure

Size

Price

Stock

Quantity

Sample (0.1mg)

In-stock

(In Japan)

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Bioz

Biological Activity

Description

A3AR antagonist 6 (Compound 5p) is a selective A₃AR antagonist with a K_i of 6.8 nM. A3AR antagonist 6 can be used in tumor research^[1].

IC₅₀ & Target^[1]

A3R

6.8 nM (Ki)

A1R

489.3 nM (Ki)

A_2AR

364 nM (Ki)

A2BR

63.6 nM (Ki)

All Adenosine Receptor Isoforms :

Chemical Information

Molecular Weight 404.44
Formula C₁₈H₂₀N₄O₅S
SMILES

O[C@@H]1[C@H](O)CS[C@H]1CN(C(N2CC3CC3)=O)C4=C(NC(C5=CC=CO5)=N4)C2=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (272 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Joung M, et al. Discovery of a Novel Template, N3‑1'-Homologated 4'-Truncated Thiosugar-Substituted Xanthine as an A3AR Antagonist via Conversion of an A1AR Antagonist. [Content Brief]

Calculators

Molarity Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Dilution Calculator

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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