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Alosetron ((Z)-2-butenedioate)

(Synonyms: GR 68755 ((Z)-2-butenedioate); GR 68755X ((Z)-2-butenedioate))
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Based on 1 publication(s) in Google Scholar

Alosetron (GR 68755) (Z)-2-butenedioate is a potent and highly selective serotonin 5-HT3 receptor antagonist. Alosetron (Z)-2-butenedioate is used for the research of irritable bowel syndrome (IBS). Alosetron (Z)-2-butenedioate blocks the fast 5HT3-mediated depolarisation of guinea-pig myenteric and submucosal neurons, with IC50 at ~55 nM. Alosetron (Z)-2-butenedioate attenuates the visceral nociceptive effect of rectal distension in conscious or anaesthetised dogs. Anti-inflammatory effects.

For research use only. We do not sell to patients.

  • CAS No.: 122852-43-1
  • Formula: C21H22N4O5
  • Molecular Weight:410.42
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • Alosetron ((Z)-2-butenedioate) Chemical Structure
    Alosetron ((Z)-2-butenedioate) Chemical Structure
CAS No.: 122852-43-1
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  • Alosetron ((Z)-2-butenedioate) Chemical Structure
    Alosetron ((Z)-2-butenedioate) Chemical Structure
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  • Alosetron ((Z)-2-butenedioate)