Arrestin-3 modulator-1
Arrestin-3 modulator-1 (Compound LSH-3) is an arrestin-3 modulator. Arrestin-3 modulator-1 binds arrestin-3 at the interdomain interface. Arrestin-3 modulator-1 enhances recruitment of arrestin-3 to phosphorylation-deficient β2AR in cells with increase of FRET levels. Arrestin-3 modulator-1 can be used for congenital disorders like retinal degeneration, hyperthyroidism and obesity research.
For research use only. We do not sell to patients.
- CAS No.: 1214645-87-0
- Formula: C24H30N4O5
- Molecular Weight:454.52
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Arrestin-3/β-Arrestin 2 |
Beta-2 adrenergic receptor |
Chemical Information
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CAS No. 1214645-87-0
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Molecular Weight 454.52
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Formula C24H30N4O5
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SMILES
CCN1CCN(C(C(O)=O)C2=CNC3=C2C=CC(NC(C4C(CC=CC4)C(O)=O)=O)=C3)CC1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)