1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor
  3. BPR1M97

BPR1M97 

Cat. No.: HY-128865 Purity: 98.99%
Handling Instructions

BPR1M97 is a dual-acting mu opioid receptor (MOP) and nociceptin-orphanin FQ peptide (NOP) receptor agonist with Ki values of 1.8 and 4.2 nM, respectively. BPR1M97 shows high potency and blood-brain barrier penetration, and produces potent antinociceptive effects.

For research use only. We do not sell to patients.

BPR1M97 Chemical Structure

BPR1M97 Chemical Structure

CAS No. : 2059904-66-2

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 269 In-stock
Estimated Time of Arrival: December 31
5 mg USD 350 In-stock
Estimated Time of Arrival: December 31
10 mg USD 550 In-stock
Estimated Time of Arrival: December 31
25 mg USD 990 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1650 In-stock
Estimated Time of Arrival: December 31
100 mg USD 2250 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

BPR1M97 is a dual-acting mu opioid receptor (MOP) and nociceptin-orphanin FQ peptide (NOP) receptor agonist with Ki values of 1.8 and 4.2 nM, respectively. BPR1M97 shows high potency and blood-brain barrier penetration, and produces potent antinociceptive effects[1].

IC50 & Target

Ki: 1.8 nM (MOP), 4.2 nM (NOP)[1]

In Vivo

BPR1M97 (1.8 mg/kg; s.c.; once) demonstrates antinociception in a murine model of cancer pain[1].

Animal Model: Male wild-type C57BL/6 mice (25-30 g)[1]
Dosage: 1.8 mg/kg
Administration: Subcutaneous injection (s.c.); once
Result: Demonstrated antinociception in a murine model of cancer pain.
Molecular Weight

349.25

Formula

C₁₈H₁₈Cl₂N₂O

CAS No.

2059904-66-2

SMILES

O=C(NCC1N(C)CCC2=C1C=CC=C2)C3=CC=C(Cl)C(Cl)=C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References
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Keywords:

BPR1M97Opioid ReceptorInhibitorinhibitorinhibit

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BPR1M97
Cat. No.:
HY-128865
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