CS-1-103
CS-1-103 is a potent estrogen receptor (ER) TRACER (transcriptional regulation via active control of epigenetic reprogramming). CS-1-103 inhibits ER transcriptional activity with an EC50 of 0.36 μM by recruiting methyl-CpG binding domain protein 2 (MBD2), HDACs and the nucleosome remodeling and deacetylase (NuRD) complex. CS-1-103 can be used for breast and prostate cancer research.
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- Formule: C41H48N6O4S
- Masse moléculaire:720.92
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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ER 0.36 μM (EC50) |
Chemical Information
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Masse moléculaire 720.92
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Formule C41H48N6O4S
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SMILES
OC1=CC=C2C(CCC3C2CC[C@@]4(C)C3CC/C4=N\OCC(NCCCCCCNC(C5=CC=CC(NC6=NC(C7=NC=CC=C7)=CS6)=C5)=O)=O)=C1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)