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Cat. No.: HY-111088

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LUF5981

LUF5981 is a relatively potent adenosine A2A receptor (A2A) antagonist with pIC₅₀ value of 6.7.

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CAS No.: 929641-63-4
Formule: C₂₄H₂₃N₃
Masse moléculaire:353.46

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

LUF5981 Chemical Structure

CAS No.: 929641-63-4

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- Cellular Effect
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
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Activité biologique

Description

LUF5981 is a relatively potent adenosine A2A receptor (A2A) antagonist with pIC₅₀ value of 6.7^[1].

Voir tous les produits spécifiques à Isoform Adenosine Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
CHO	IC₅₀	1.7 μM Compound: 14, LUF 5981	Activity at human adenosine A1 receptor in CHO cells assessed as effect on CPA induced inhibition of forskolin-stimulated cAMP production Activity at human adenosine A1 receptor in CHO cells assessed as effect on CPA induced inhibition of forskolin-stimulated cAMP production	[PMID: 17300165]

Chemical Information

CAS No. 929641-63-4
Masse moléculaire 353.46
Formule C₂₄H₂₃N₃
SMILES

C12=NC(C3=CC=CC=C3)=CC(C4=CC=CC=C4)=C1N=C(C5CCCCC5)N2
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (268 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Fan Fan, et al. The integration of pharmacophore-based 3D QSAR modeling and virtual screening in safety profiling: A case study to identify antagonistic activities against adenosine receptor, A2A, using 1,897 known drugs. PLoS One. 2019 Jan 3;14(1):e0204378. [Content Brief]

Calculators

Calculateur de molarité

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Calculateur de dilution

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Activité biologique
- Description
Chemical Information
Pureté et documentation
Références

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LUF5981

Voir tous les produits spécifiques à Isoform Adenosine Receptor

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

LUF5981 Related Classifications

HY-111088 Related Classifications