2819989-75-6
2819989-75-6
Chemical Structure
PBRM1-BD2-IN-8
- CAS No.: 2819989-75-6
- Formula:C15H13BrN2O
- Molecular Weight:317.18
IUPAC Name: 5-hydroxybenzo[d]oxazol-2(3H)-one
InChIKey: PXWIXTCIXZCREB-UHFFFAOYSA-N
SMILES: O=C1NC(C2=CC=CC(C)=C2)NC3=C1C(Br)=CC=C3
Biological Activity: PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor (PBRM1-BD2 Kd=4.4 μM, PBRM1-BD2 IC50=0.16 μM; PBRM1-BD5 Kd=25 μM). PBRM1-BD2-IN-8 shows anti-cancer activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PBRM1-BD2-IN-8 | 98.05% | PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor (PBRM1-BD2 Kd=4.4 μM, PBRM1-BD2 IC50=0.16 μM; PBRM1-BD5 Kd=25 μM). PBRM1-BD2-IN-8 shows anti-cancer activity. | ||||||||||||||||||||
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References
Keywords
