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Cat. No.: HY-118014

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CAY10535

Name: CAY10535
Brand: MedChemExpress
SKU: HY-118014
Price: 79.00 USD
Availability: InStock
Rating: 5 (1 reviews)

CAY10535 is a FP and TP receptor inhibitor and can be used for research of cardiovascular diseases.

Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.

CAS No.: 945716-28-9
Formule: C₁₈H₂₁N₃O₇S
Masse moléculaire:423.44

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

CAY10535 Chemical Structure

CAS No.: 945716-28-9

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
- Cellular Effect
- In Vitro
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

CAY10535 is a FP and TP receptor inhibitor and can be used for research of cardiovascular diseases^[1].

IC₅₀ & Target

TP Receptor

FP Receptor

Voir tous les produits spécifiques à Isoform Prostaglandin Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
HEK293	IC₅₀	1970 nM Compound: 9ag	Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobilization Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobilization	[PMID: 17630727]
HEK293	IC₅₀	99 nM Compound: 9ag	Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobilization Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobilization	[PMID: 17630727]

In Vitro

CAY10535 (10 μM) significantly inhibits PGF_2α (1 μM) and/or capsaicin (2 μM) induced coronary rings contractions^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 945716-28-9
Masse moléculaire 423.44
Formule C₁₈H₂₁N₃O₇S
SMILES

O=S(C1=CC([N+]([O-])=O)=CC=C1OC2=CC=CC(OC)=C2)(NC(NC(C)(C)C)=O)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. S Christopher Hiett, et al. Mechanisms underlying capsaicin effects in canine coronary artery: implications for coronary spasm. Cardiovasc Res. 2014 Sep 1;103(4):607-18. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

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