XH-30
XH-30 is a potent, selective, and orally active PKMYT1 inhibitor, with an IC50 of 4.1 nM. XH-30 suppresses the proliferation of P53-mutated triple-negative breast cancer (TNBC) cells by inducing G2/M phase release, DNA damage, and apoptosis. XH-30 demonstrates antitumor effects in an MDA-MB-231 mouse model. XH-30 can be used for P53-mutated TNBC research.
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- CAS. Nr.: 3077136-87-6
- Formel: C19H19N3O3
- Molecular Weight:337.37
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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PKMYT1 4.1 nM (IC50) |
Chemical Information
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CAS. Nr. 3077136-87-6
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Molecular Weight 337.37
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Formel C19H19N3O3
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SMILES
NC1=C(C=C2N=C(OC2=C1C3=C(C(O)=CC=C3C)C)C4CC4)C(N)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
XH-30 Related Classifications
HY-180893 Related Classifications
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