OMDM-1
Based on 1 Customer Validation
OMDM-1 is a potent, selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 2.4 μM.
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- Pureté: 98.05%
- CAS No.: 616884-62-9
- Formule: C27H45NO3
- Masse moléculaire:431.65
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Stockage:
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
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Solvant et solubilité
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
Ki: 2.4 μM (anandamide cellular uptake)[1]
OMDM-1 shows poor affinity for either CB1 (Ki=12.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively; OMDM-1 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50≥10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 616884-62-9
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Appearance Solid
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Masse moléculaire 431.65
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Formule C27H45NO3
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Color White to off-white
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SMILES
CCCCCCCC/C=C\CCCCCCCC(N[C@@H](CC1=CC=C(O)C=C1)CO)=O
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Structure Classification
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Initial Source
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Solvant et solubilité
DMSO : 100 mg/mL (231.67 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pureté et documentation
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Fiche technique (266 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Instruction de manipulation (2659 KB)
Références
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.3167 mL | 11.5835 mL | 23.1669 mL | 57.9173 mL |
| 5 mM | 0.4633 mL | 2.3167 mL | 4.6334 mL | 11.5835 mL | |
| 10 mM | 0.2317 mL | 1.1583 mL | 2.3167 mL | 5.7917 mL | |
| 15 mM | 0.1544 mL | 0.7722 mL | 1.5445 mL | 3.8612 mL | |
| 20 mM | 0.1158 mL | 0.5792 mL | 1.1583 mL | 2.8959 mL | |
| 25 mM | 0.0927 mL | 0.4633 mL | 0.9267 mL | 2.3167 mL | |
| 30 mM | 0.0772 mL | 0.3861 mL | 0.7722 mL | 1.9306 mL | |
| 40 mM | 0.0579 mL | 0.2896 mL | 0.5792 mL | 1.4479 mL | |
| 50 mM | 0.0463 mL | 0.2317 mL | 0.4633 mL | 1.1583 mL | |
| 60 mM | 0.0386 mL | 0.1931 mL | 0.3861 mL | 0.9653 mL | |
| 80 mM | 0.0290 mL | 0.1448 mL | 0.2896 mL | 0.7240 mL | |
| 100 mM | 0.0232 mL | 0.1158 mL | 0.2317 mL | 0.5792 mL |
OMDM-1 Related Classifications
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