OMDM-4
OMDM-4 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki 17.7 μM.
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- CAS No.: 616884-65-2
- Formule: C29H43NO3
- Masse moléculaire:453.66
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
Ki: 17.7 μM (anandamide cellular uptake)[1]
OMDM-4 shows poor affinity for either CB1 (Ki=4.9 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively. OMDM-4 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50>10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 616884-65-2
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Masse moléculaire 453.66
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Formule C29H43NO3
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SMILES
CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(N[C@H](CC1=CC=C(O)C=C1)CO)=O
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Structure Classification
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Initial Source
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
OMDM-4 Related Classifications
HY-135880A Related Classifications
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