ERK5-IN-6
ERK5-IN-6 (compound 5J) is an ERK5 kinase inhibitor with anticancer activity. ERK5-IN-6 exhibits good anti-proliferative activity with the IC50 value of 4.56 µg/mL for A549 cells.
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- CAS No.: 2734916-64-2
- Formule: C23H21N3
- Masse moléculaire:339.43
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
|
ERK |
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| A549 | IC50 |
4.56 μg/mL
Compound: 5j
|
Antiproliferative activity against human A549 cells assessed as cell growth inhibition incubated for 48 hrs by MTT assay
Antiproliferative activity against human A549 cells assessed as cell growth inhibition incubated for 48 hrs by MTT assay
|
[PMID: 37862935] |
Chemical Information
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CAS No. 2734916-64-2
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Masse moléculaire 339.43
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Formule C23H21N3
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SMILES
C12=NC=CC=C1C(C3=CCN(CC4=CC=C5C=CC=CC5=C4)CC3)=CN2
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Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)