ERK5-IN-6
ERK5-IN-6 (compound 5J) is an ERK5 kinase inhibitor with anticancer activity. ERK5-IN-6 exhibits good anti-proliferative activity with the IC50 value of 4.56 µg/mL for A549 cells.
For research use only. We do not sell to patients.
- CAS No.: 2734916-64-2
- Formula: C23H21N3
- Molecular Weight:339.43
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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ERK |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| A549 | IC50 |
4.56 μg/mL
Compound: 5j
|
Antiproliferative activity against human A549 cells assessed as cell growth inhibition incubated for 48 hrs by MTT assay
Antiproliferative activity against human A549 cells assessed as cell growth inhibition incubated for 48 hrs by MTT assay
|
[PMID: 37862935] |
Chemical Information
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CAS No. 2734916-64-2
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Molecular Weight 339.43
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Formula C23H21N3
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SMILES
C12=NC=CC=C1C(C3=CCN(CC4=CC=C5C=CC=CC5=C4)CC3)=CN2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)