MRS1177
MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 183721-13-3
- Fòrmula: C20H12ClN5O2
- Peso molecular:389.79
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
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Actividad biológica
Chemical Information
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No. CAS 183721-13-3
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Peso molecular 389.79
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Fòrmula C20H12ClN5O2
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SMILES
O=C(C1=CC=CC=C1)NC2=NC3=C(C4=NC(C5=CC=CO5)=NN24)C=C(C=C3)Cl
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
[1]. Tafi A, et al. Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. J Med Chem. 2006 Jul 13;49(14):4085-97. [Content Brief]
[2]. Cheong SL, et al. Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo-pyrimidines as potent human A3 adenosine receptor antagonists. Bioorg Med Chem Lett. 2011 May 15;21(10):2898-905. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MRS1177 Related Classifications
HY-120090 Related Classifications
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