Pexopiprant
Based on 1 Customer Validation
Pexopiprant is an oral antagonist of the prostaglandin D2 receptor 2 (DP2),Ki ＜ 100nM. Pexopiprant can be used in studies of asthma.
Para uso exclusivo en investigación. No vendemos a pacientes.
- Pureza : 99.40%
- No. CAS: 932708-14-0
- Fòrmula: C21H17Cl2F2NO4
- Peso molecular:456.27
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Almacenamiento:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Actividad biológica
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Chemical Information
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Solvente y solubilidad
- Pureza y Documentación
- Referencias
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Help & FAQs
Actividad biológica
Descripciòn
IC50 & Target
[1]|
DP2 <100 nM (Ki) |
Chemical Information
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No. CAS 932708-14-0
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Appearance Solid
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Peso molecular 456.27
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Fòrmula C21H17Cl2F2NO4
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Color Off-white to light yellow
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SMILES
O=C(O)COC1=C2C(OC(F)F)=C(CC3=CC=C(Cl)C=C3)C(CC)=NC2=C(Cl)C=C1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvente y solubilidad
In Vitro:
DMSO : 100 mg/mL (219.17 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pureza y Documentación
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Ficha de datos (273 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Instrucciones de manejo (2659 KB)
Referencias
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.1917 mL | 10.9584 mL | 21.9168 mL | 54.7921 mL |
| 5 mM | 0.4383 mL | 2.1917 mL | 4.3834 mL | 10.9584 mL | |
| 10 mM | 0.2192 mL | 1.0958 mL | 2.1917 mL | 5.4792 mL | |
| 15 mM | 0.1461 mL | 0.7306 mL | 1.4611 mL | 3.6528 mL | |
| 20 mM | 0.1096 mL | 0.5479 mL | 1.0958 mL | 2.7396 mL | |
| 25 mM | 0.0877 mL | 0.4383 mL | 0.8767 mL | 2.1917 mL | |
| 30 mM | 0.0731 mL | 0.3653 mL | 0.7306 mL | 1.8264 mL | |
| 40 mM | 0.0548 mL | 0.2740 mL | 0.5479 mL | 1.3698 mL | |
| 50 mM | 0.0438 mL | 0.2192 mL | 0.4383 mL | 1.0958 mL | |
| 60 mM | 0.0365 mL | 0.1826 mL | 0.3653 mL | 0.9132 mL | |
| 80 mM | 0.0274 mL | 0.1370 mL | 0.2740 mL | 0.6849 mL | |
| 100 mM | 0.0219 mL | 0.1096 mL | 0.2192 mL | 0.5479 mL |
Pexopiprant Related Classifications
HY-109186 Related Classifications
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