GPR30 agonist-1
Based on 1 Customer Validation
GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects.
For research use only. We do not sell to patients.
- Purity: 98.62%
- CAS No.: 415919-74-3
- Formula: C19H17BrFNO
- Molecular Weight:374.25
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 415919-74-3
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Appearance Solid
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Molecular Weight 374.25
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Formula C19H17BrFNO
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Color White to off-white
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SMILES
COC(C=C1)=C(C=C1Br)[C@@]2([H])[C@](CC=C3)([H])[C@]3([H])C4=CC(F)=CC=C4N2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 50 mg/mL (133.60 mM; ultrasonic and warming and heat to 80°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (273 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.6720 mL | 13.3601 mL | 26.7201 mL | 66.8003 mL |
| 5 mM | 0.5344 mL | 2.6720 mL | 5.3440 mL | 13.3601 mL | |
| 10 mM | 0.2672 mL | 1.3360 mL | 2.6720 mL | 6.6800 mL | |
| 15 mM | 0.1781 mL | 0.8907 mL | 1.7813 mL | 4.4534 mL | |
| 20 mM | 0.1336 mL | 0.6680 mL | 1.3360 mL | 3.3400 mL | |
| 25 mM | 0.1069 mL | 0.5344 mL | 1.0688 mL | 2.6720 mL | |
| 30 mM | 0.0891 mL | 0.4453 mL | 0.8907 mL | 2.2267 mL | |
| 40 mM | 0.0668 mL | 0.3340 mL | 0.6680 mL | 1.6700 mL | |
| 50 mM | 0.0534 mL | 0.2672 mL | 0.5344 mL | 1.3360 mL | |
| 60 mM | 0.0445 mL | 0.2227 mL | 0.4453 mL | 1.1133 mL | |
| 80 mM | 0.0334 mL | 0.1670 mL | 0.3340 mL | 0.8350 mL | |
| 100 mM | 0.0267 mL | 0.1336 mL | 0.2672 mL | 0.6680 mL |