1. GPCR/G Protein
  2. Free Fatty Acid Receptor
  3. GPR40/FFAR1 modulator 1

GPR40/FFAR1 modulator 1 

Cat. No.: HY-111763 Purity: 99.11%
Handling Instructions

GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1).

For research use only. We do not sell to patients.

GPR40/FFAR1 modulator 1 Chemical Structure

GPR40/FFAR1 modulator 1 Chemical Structure

CAS No. : 874755-26-7

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Free Sample (0.5-1 mg)   Apply Now  
5 mg USD 55 In-stock
Estimated Time of Arrival: December 31
10 mg USD 90 In-stock
Estimated Time of Arrival: December 31
25 mg USD 160 In-stock
Estimated Time of Arrival: December 31
50 mg USD 260 In-stock
Estimated Time of Arrival: December 31
100 mg USD 420 In-stock
Estimated Time of Arrival: December 31
500 mg USD 850 In-stock
Estimated Time of Arrival: December 31
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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1)[1].

IC50 & Target

Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1)[1].

Molecular Weight

389.41

Formula

C21H19N5O3

CAS No.
SMILES

CC1=CC=CC=C1NC2=NC(COC3=CC=C(C(C)=CC(O4)=O)C4=C3)=NC(N)=N2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Solvent & Solubility
In Vitro: 

DMSO : 31.25 mg/mL (80.25 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5680 mL 12.8399 mL 25.6799 mL
5 mM 0.5136 mL 2.5680 mL 5.1360 mL
10 mM 0.2568 mL 1.2840 mL 2.5680 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.08 mg/mL (5.34 mM); Clear solution

*All of the co-solvents are available by MCE.
Purity & Documentation
References
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
GPR40/FFAR1 modulator 1
Cat. No.:
HY-111763
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