LUF5981
LUF5981 is a relatively potent adenosine A2A receptor (A2A) antagonist with pIC50 value of 6.7.
For research use only. We do not sell to patients.
- CAS No.: 929641-63-4
- Formula: C24H23N3
- Molecular Weight:353.46
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adenosine Receptor Isoforms
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Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
1.7 μM
Compound: 14, LUF 5981
|
Activity at human adenosine A1 receptor in CHO cells assessed as effect on CPA induced inhibition of forskolin-stimulated cAMP production
Activity at human adenosine A1 receptor in CHO cells assessed as effect on CPA induced inhibition of forskolin-stimulated cAMP production
|
[PMID: 17300165] |
Chemical Information
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CAS No. 929641-63-4
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Molecular Weight 353.46
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Formula C24H23N3
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SMILES
C12=NC(C3=CC=CC=C3)=CC(C4=CC=CC=C4)=C1N=C(C5CCCCC5)N2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)