FFA2 agonist-2
FFA2 agonist-2 is a potent agonist of the FFA2 (GPR43) receptor, with a pEC50 of 7.9 for human FFA2, and a pEC50 of 7.3 for murine FFA2. FFA2 agonist-2 acts as an orthosteric agonist and shows no obvious cross‑activity against FFA1, FFA3 and FFA4. FFA2 agonist-2 can be used for FFA2 receptor research in type 2 diabetes and metabolic disorders.
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- CAS 番号: 1229363-11-4
- 分子式: C23H20Cl2N2O3S
- 分子量:475.39
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- プロトコル
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
製品説明
IC50 & Target
[1]|
FFAR2 7.9 (pEC50, 人源) |
FFAR2 7.3 (pEC50, 鼠源) |
体外実験
FFA2 agonist-2 (compound 8) acts as a potent agonist at both hFFA2 and mFFA2 receptors in CHO cells, with a pEC50 of 7.9 (hFFA2) and 7.3 (mFFA2), and binds to hFFA2 with a pKi of 6.7[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Parmacokinetics
体内実験
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 1229363-11-4
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分子量 475.39
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分子式 C23H20Cl2N2O3S
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SMILES
OC(C[C@@H](CC1=CC=CC=C1)C(N(C2CC2)C3=NC(C4=C(C=CC(Cl)=C4)Cl)=CS3)=O)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
FFA2 agonist-2 関連分類
HY-182729 関連分類
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