OMDM-1
Based on 1 Customer Validation
OMDM-1 is a potent, selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 2.4 μM.
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- 純度: 98.05%
- CAS 番号: 616884-62-9
- 分子式: C27H45NO3
- 分子量:431.65
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保管条件:
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
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Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
Endogenous Metabolite アイソフォーム固有の製品をすべて表示
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生物活性
Ki: 2.4 μM (anandamide cellular uptake)[1]
OMDM-1 shows poor affinity for either CB1 (Ki=12.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively; OMDM-1 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50≥10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 616884-62-9
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性状 Solid
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分子量 431.65
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分子式 C27H45NO3
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Color White to off-white
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SMILES
CCCCCCCC/C=C\CCCCCCCC(N[C@@H](CC1=CC=C(O)C=C1)CO)=O
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Structure Classification
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Initial Source
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
溶剤 & 溶解度
DMSO : 100 mg/mL (231.67 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (266 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.3167 mL | 11.5835 mL | 23.1669 mL | 57.9173 mL |
| 5 mM | 0.4633 mL | 2.3167 mL | 4.6334 mL | 11.5835 mL | |
| 10 mM | 0.2317 mL | 1.1583 mL | 2.3167 mL | 5.7917 mL | |
| 15 mM | 0.1544 mL | 0.7722 mL | 1.5445 mL | 3.8612 mL | |
| 20 mM | 0.1158 mL | 0.5792 mL | 1.1583 mL | 2.8959 mL | |
| 25 mM | 0.0927 mL | 0.4633 mL | 0.9267 mL | 2.3167 mL | |
| 30 mM | 0.0772 mL | 0.3861 mL | 0.7722 mL | 1.9306 mL | |
| 40 mM | 0.0579 mL | 0.2896 mL | 0.5792 mL | 1.4479 mL | |
| 50 mM | 0.0463 mL | 0.2317 mL | 0.4633 mL | 1.1583 mL | |
| 60 mM | 0.0386 mL | 0.1931 mL | 0.3861 mL | 0.9653 mL | |
| 80 mM | 0.0290 mL | 0.1448 mL | 0.2896 mL | 0.7240 mL | |
| 100 mM | 0.0232 mL | 0.1158 mL | 0.2317 mL | 0.5792 mL |
OMDM-1 関連分類
HY-121557 関連分類
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