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Cat. No.: HY-118678

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MRS1186

MRS1186 is a potent and selective human Adenosine A3 receptor (hA₃AR) antagonist, with a K_i of 7.66 nM.

연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.

CAS No.: 183721-03-1
화학식: C₁₆H₁₂ClN₅O₂
분자량:341.75

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

MRS1186 Chemical Structure

CAS No.: 183721-03-1

Amount: USD 0.00

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- IC₅₀ & Target
- In Vitro
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

제품 설명

MRS1186 is a potent and selective human Adenosine A3 receptor (hA₃AR) antagonist, with a K_i of 7.66 nM.

IC₅₀ & Target

Ki: 7.66 nM (hA₃AR)^[1].

All Adenosine Receptor Isoforms :

In Vitro

MRS1186 (compound 2d) is a potent and selective human Adenosine A3 receptor (hA₃AR) antagonist, with a K_i of 7.66 nM^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 183721-03-1
분자량 341.75
화학식 C₁₆H₁₂ClN₅O₂
SMILES

CCC(NC1=NC2=C(C3=NC(C4=CC=CO4)=NN13)C=C(C=C2)Cl)=O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Tafi A, et al. Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. J Med Chem. 2006 Jul 13;49(14):4085-97. [Content Brief]

Calculators

몰농도 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

농도 희석 계산기

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

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Other size

견적 받기

Amount: USD 0.00

Biological Activity
- 제품 설명
- IC₅₀ & Target
- In Vitro
Chemical Information
순도&문서
References

상품명:
Cat. No.:
수량:
MCE Japan Authorized Agent:

상품명:
CAS No.:
Species:
Purity:
수량:

MRS1186

DPCPX

CGS 21680

CGS 21680 Hydrochloride

Piclidenoson

Ciforadenant

Namodenoson

Derenofylline

CGS 15943

GR79236

Capadenoson

Rolofylline

Proxyphylline

All Adenosine Receptor Isoforms

Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

Bioz

MRS1186

DPCPX

CGS 21680

CGS 21680 Hydrochloride

Piclidenoson

Ciforadenant

Namodenoson

Derenofylline

CGS 15943

GR79236

Capadenoson

Rolofylline

Proxyphylline

All Adenosine Receptor Isoforms

Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

MRS1186 Related Classifications

HY-118678 Related Classifications

Bioz