Biphalin TFA
Biphalin TFA, a BBB-penetrable opioid peptide analog, contains two active enkephalin pharmacophores. Biphalin TFA has high affinity for opioid receptors. Biphalin TFA shows analgesic effect in acute, neuropathic, and chronic animal pain models. Biphalin TFA is also an antiviral, antiproliferative, anti-inflammatory, and neuroprotective agent.
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- CAS No.: 126872-95-5
- 화학식: C46H56N10O10·xC2HF3O2
- 분자량:909.00 (free base)
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Opioid Receptor Isoforms
More
Biological Activity
Chemical Information
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CAS No. 126872-95-5
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분자량 909.00 (free base)
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화학식 C46H56N10O10·xC2HF3O2
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Sequence
Tyr-{dAla}-Gly-Phe-NH2 (covalent bridge:Phe-Phe, dimer)
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Sequence Shortening
Y-{D-Ala}-GF-NH2 (covalent bridge:Phe-Phe, dimer)
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
[1]. T J Abbruscato, et al. Blood-to-central nervous system entry and stability of biphalin, a unique double-enkephalin analog, and its halogenated derivatives. J Pharmacol Exp Ther. 1996, 276,3. [Content Brief]
[2]. Redkiewicz P, et al. Biphalin-A Potent Opioid Agonist-As a Panacea for Opioid System-Dependent Pathophysiological Diseases? Int J Mol Sci. 2021 Oct 21;22(21):11347. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)