LSD1/2-IN-4
LSD1/2-IN-4, a PCPA derivative, is an inhibitor of lysine-specific demethylase 1 (LSD1) and lysine-specific demethylase 2 (LSD2). LSD1/2-IN-4 inhibits LSD1 and LSD2 with Ki values of 0.11 μM and 130 μM, respectively. LSD1/2-IN-4 can be used for the research of several cancers including T-cell acute lymphoblastic leukemia (TALL).
For research use only. We do not sell to patients.
- CAS No.: 2821068-09-9
- Formula: C9H8BrF2N
- Molecular Weight:248.07
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
KDM1/LSD1 |
LSD1/2-IN-4 shows strong inhibitory activity against both LSD1 and LSD2 with Ki values of 0.11 μM and 130 μM, respectively and not inhibits peroxidase with an IC50 >500 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS No. 2821068-09-9
-
Molecular Weight 248.07
-
Formula C9H8BrF2N
-
SMILES
N[C@@H]1C[C@H]1C2=CC(F)=C(Br)C(F)=C2
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LSD1/2-IN-4 Related Classifications
HY-151194 Related Classifications
Powered by Bioz