LSD1-IN-16
LSD1-IN-16 (compound 4b) is a potent LSD1 inhibitor. LSD1-IN-16 can inhibit LSD1-CoREST, MAO-A and MAO-B, with IC50 values of 0.015, 0.024, and 0.366 μM, respectively. LSD1-IN-16 displays cell growth arrest in prostate cancer LNCaP cells, with an IC50 of 15.2 μM.
For research use only. We do not sell to patients.
- CAS No.: 3033060-68-0
- Formula: C20H18N2OS
- Molecular Weight:334.43
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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KDM1/LSD1 |
MAO-A 0.024 ± μM (IC50) |
MAO-B 0.366 ± μM (IC50) |
Chemical Information
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CAS No. 3033060-68-0
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Molecular Weight 334.43
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Formula C20H18N2OS
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SMILES
NC1CC1C2=CC=C(C=C2)NC(C3=CC=CC(C4=CC=CS4)=C3)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)