mAChR-IN-1
mAChR-IN-1 is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM.
For research use only. We do not sell to patients.
- CAS No.: 119391-56-9
- Formula: C23H25IN2O2
- Molecular Weight:488.36
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
Biological Activity
Chemical Information
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CAS No. 119391-56-9
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Appearance Solid
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Molecular Weight 488.36
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Formula C23H25IN2O2
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Color White to off-white
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SMILES
O=C(C(C1CCN(CC2=CC=C(I)C=C2)CC1)(C3=CC=CC=C3)CC4)NC4=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year
Solvent & Solubility
DMSO : ≥ 52 mg/mL (106.48 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (274 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.0477 mL | 10.2383 mL | 20.4767 mL | 51.1917 mL |
| 5 mM | 0.4095 mL | 2.0477 mL | 4.0953 mL | 10.2383 mL | |
| 10 mM | 0.2048 mL | 1.0238 mL | 2.0477 mL | 5.1192 mL | |
| 15 mM | 0.1365 mL | 0.6826 mL | 1.3651 mL | 3.4128 mL | |
| 20 mM | 0.1024 mL | 0.5119 mL | 1.0238 mL | 2.5596 mL | |
| 25 mM | 0.0819 mL | 0.4095 mL | 0.8191 mL | 2.0477 mL | |
| 30 mM | 0.0683 mL | 0.3413 mL | 0.6826 mL | 1.7064 mL | |
| 40 mM | 0.0512 mL | 0.2560 mL | 0.5119 mL | 1.2798 mL | |
| 50 mM | 0.0410 mL | 0.2048 mL | 0.4095 mL | 1.0238 mL | |
| 60 mM | 0.0341 mL | 0.1706 mL | 0.3413 mL | 0.8532 mL | |
| 80 mM | 0.0256 mL | 0.1280 mL | 0.2560 mL | 0.6399 mL | |
| 100 mM | 0.0205 mL | 0.1024 mL | 0.2048 mL | 0.5119 mL |