MerTK/Axl-IN-1
MerTK/Axl-IN-1 (Compound A-910) is a potent and selective dual MerTK/Axl inhibitor, with IC50s of 4.2 and 8.8 nM in Ba/F3, and 0.2 and 0.9 nM in HTRF. MerTK/Axl-IN-1 results in pMerTK inhibition in vivo. MerTK/Axl-IN-1 has long half-life, high oral exposure and bioavailability.
For research use only. We do not sell to patients.
- CAS No.: 3036009-40-9
- Formula: C40H47FN6O4
- Molecular Weight:694.84
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Chemical Information
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CAS No. 3036009-40-9
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Molecular Weight 694.84
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Formula C40H47FN6O4
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SMILES
FC1=NC=CC=C1C2=CC(C(N[C@H]3CCC[C@@H]3OCC4=CC=C(C5=CC(CCC[C@@H]6N7CCN(C[C@@H](CO)O)CC7)=C6C=C5)C=C4)=O)=C(N)N=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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