country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-P10761A

Copy Link Print Information

NOTA-DPI-4452 TFA

Name: NOTA-DPI-4452 TFA
Brand: MedChemExpress
SKU: HY-P10761A
Price: 460.00 USD
Availability: InStock
Rating: 5 (1 reviews)

Customer Review

Based on 1 Customer Validation

NOTA-DPI-4452 TFA is a trifluoroacetate derivative with DPI-4452 (HY-P10761) as the parent peptide. DPI-4452 is a CAIX-targeting cyclic peptide with a DOTA cage that can chelate with radionuclides and is used to express CAIX tumors for PET-CT imaging and research.

For research use only. We do not sell to patients.

Formula: C₈₈H₁₂₅N₂₁O₂₇S₃·xC₂HF₃O₂
Molecular Weight:2005.25 (free base)

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

NOTA-DPI-4452 TFA Chemical Structure

Size

Price

Stock

Quantity

Amount: USD 0.00

* Please select Quantity before adding items.

Top Publications Citing

Use of MCE Products

One-stop CDMO Service

One-Stop Platform：From Independent R&D to Pilot-Scale Production

Biological Activity
- Description
- In Vitro
Chemical Information
Solvent & Solubility
- In Vitro
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

All Radionuclide-Drug Conjugates (RDCs) Isoforms :

All Carbonic Anhydrase Isoforms :

In Vitro

NOTA-DPI-4452 TFA is a trifluoroacetate derivative with DPI-4452 (HY-P10761) as the parent peptide^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

Molecular Weight 2005.25 (free base)
Formula C₈₈H₁₂₅N₂₁O₂₇S₃·xC₂HF₃O₂
SMILES

C[C@@H](O)[C@H](NC([C@@H](N1)CC(C)C)=O)C(N[C@@H](CC2=CNC3=C2C=CC=C3)C(N[C@H](C(N[C@@H](CSCC4=CC(CSC[C@H](NC([C@@H](NC(CN5CCN(C(CN6CCN(CC(O)=O)CCN(CC(O)=O)CC6)=O)CC5)=O)CCC(N)=O)=O)C(N[C@@H](CCC(O)=O)C(N(CCC7)[C@H]7C(N[C@@H](CC(O)=O)C(N[C@@H](CC8=CC=CC(NC(CCCS(=O)(N)=O)=O)=C8)C1=O)=O)=O)=O)=O)=CC=C4)C(N)=O)=O)CO)=O)=O.OC(C(F)(F)F)=O.[x]
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Solvent & Solubility

In Vitro:

DMSO : 100 mg/mL (Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

View the Complete Stock Solution Preparation Table

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Massière, et al. Preclinical Characterization of DPI-4452: A68Ga/177Lu Theranostic Ligand for Carbonic Anhydrase IX. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2024, 65(5), 761–767. [Content Brief]

Calculators

Molarity Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Dilution Calculator

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

Get Quote In-stock

Other size

Get Quote