1. Metabolic Enzyme/Protease
  2. Endogenous Metabolite
  3. OMDM-2

OMDM-2 

Cat. No.: HY-103342
Handling Instructions

OMDM-2 is a potent, selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 3.0 μM.

For research use only. We do not sell to patients.

OMDM-2 Chemical Structure

OMDM-2 Chemical Structure

CAS No. : 616884-63-0

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Description

OMDM-2 is a potent, selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 3.0 μM[1].

IC50 & Target

Ki: 3.0 μM (anandamide cellular uptake)[1]

In Vitro

OMDM-2 shows poor affinity for either CB1 (Ki=5.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively; OMDM-2 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50=10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].

Molecular Weight

431.65

Formula

C₂₇H₄₅NO₃

CAS No.

616884-63-0

SMILES

CCCCCCCC/C=C\CCCCCCCC(N[[email protected]](CC1=CC=C(O)C=C1)CO)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

OMDM-2OMDM2OMDM 2Endogenous MetabolitefattyacidsuptakeRBL-2H3cellsvanilloidVR1cannabinoidreceptortype1CB1CB2FAAHInhibitorinhibitorinhibit

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