2. PROTAC Cell Cycle/DNA Damage
  3. PROTACs SWI/SNF Complex
  4. PROTAC SMARCA2 degrader-32

PROTAC SMARCA2 degrader-32 (Compound 27) is the degrader for SMARCA2 with a DC50 of 1.3 nM. PROTAC SMARCA2 degrader-32 inhibits the proliferation of lung cancer cell NCI-H838 with a GI50 of 34 nM. (Pink: ligand for target protein SMARCA2 ligand-11 (HY-170349); Black: linker (HY-W895794); Blue: ligand for E3 ligase VHL (HY-170348))

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PROTAC SMARCA2 degrader-32

PROTAC SMARCA2 degrader-32 화학구조

CAS No. : 3033586-50-1

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PROTAC SMARCA2 degrader-32 Related Antibodies

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제품 설명

PROTAC SMARCA2 degrader-32 (Compound 27) is the degrader for SMARCA2 with a DC50 of 1.3 nM. PROTAC SMARCA2 degrader-32 inhibits the proliferation of lung cancer cell NCI-H838 with a GI50 of 34 nM[1]. (Pink: ligand for target protein SMARCA2 ligand-11 (HY-170349); Black: linker (HY-W895794); Blue: ligand for E3 ligase VHL (HY-170348))

분자량

970.66

화학식

C54H64ClN9O4S
CAS No.
SMILES

CC1(C(N(C2=CC=CC(Cl)=C23)C4=CC(C5CCN(CC5)C[C@@H]6CC[C@@H](C7=CN(N=N7)[C@@H](C(C)(C)C)C(N8[C@@H](C[C@H](C8)O)C(N[C@H](C9=CC=C(C%10=C(N=CS%10)C)C=C9)C)=O)=O)CC6)=CC=C41)=NC3=O)C
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
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PROTAC SMARCA2 degrader-32 Related Classifications

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Keywords:

PROTAC SMARCA2 degrader-323033586-50-1PROTACsSWI/SNF ComplexSWI/SNF Family of Chromatin-Remodelling ComplexesNCI-H838Calu-6HT1080Inhibitorinhibitorinhibit

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상품명:
PROTAC SMARCA2 degrader-32
Cat. No.:
HY-170343
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