346 Results for "

low affinity

" in MedChemExpress (MCE) Product Catalog:
Products (346)

346 Results for "low affinity" in MCE Product Catalog:

Cat. No.: HY-14945
CAS No.: 442201-24-3
Purity:  99.81%
Synonyms: GSK189075
Target:  

SGLT

Research Areas:  

Metabolic Disease

Remogliflozin etabonate (GSK189075) is an orally active, selective and low-affinity sodium glucose cotransporter (SGLT2) inhibitor with Ki values of 1.95 μM, 2.14 μM, 43.1 μM, 8.57 μM for hSGLT2, rSGLT2, hSGLT1, rSGLT1, respectively. Remogliflozin etabonate is a proagent based on benzylpyrazole glucoside and is metabolized to its active form, Remogliflozin, in the body. Remogliflozin etabonate exhibits antidiabetic efficacy in rodent models .
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Cat. No.: HY-173043
Target:  

5-HT Receptor

Research Areas:  

Cancer

5-HT6R antagonist 6 exhibits high affinity and selectivity for 5-HT6R , with a Ki value of 42 nM. 5-HT6R antagonist 6 shows weak antiproliferative activity against tumor cells and low toxicity to normal cells. 5-HT6R antagonist 6 can be used in the study of cancer .
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Cat. No.: HY-184780
CAS No.: 84731-70-4
Research Areas:  

Others

Eco-DEHCH is a phthalate-free alternative plasticizer that safely and effectively softens plastics such as flexible PVC. Eco-DEHCH shows low binding affinity for various endocrine receptors, including estrogen, androgen, glucocorticoid, thyroid receptor α and thyroid receptor β. Eco-DEHCH causes dose-dependent accumulation of α2u-globulin in the kidneys of male Han Wistar rats, but has overall general safety .
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Cat. No.: HY-P991749

Target:  

Interleukin Related

Research Areas:  

Inflammation/Immunology

Anti-Rat CD25 Antibody (OX-39) recognizes the 55 kDa low-affinity interleukin-2 receptor α chain (IL-2R α, CD25). Anti-Rat CD25 Antibody (OX-39) interacts with a single class of sites on the alpha chain of the rat R-IL2 with a high affinity (Kd of 0.8 nM) and competes with IL2 binding on this chain (Ki of 0.53 nM). Anti-Rat CD25 Antibody (OX-39) is a weak inhibitor in vitro on IL2-induced proliferation and in vivo on allograft rejection. Recommend Isotype Controls: Mouse IgG1 kappa, Isotype Control (HY-P99977) .
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Cat. No.: HY-P7271
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: NGFR; low affinity Neurotrophin Receptor P75NTR; Nerve Growth Factor Receptor; TNFR Superfamily, Member 16; TNFRSF16; NGF Receptor; P75NTR; Gp80-LNGFR; CD271; P75 ICD; Tumor Necrosis Factor Receptor Superfamily Member 16; Nerve Growth Factor Receptor (TNF
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P7783
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: CSF2RA; GMCSFR-Alpha; Prev. CSF2R; CDw116; AlphaGMR; CSF2RY; CD116; Granulocyte-Macrophage Colony-Stimulating Factor Receptor Alpha Chain; Colony Stimulating Factor 2 Receptor, Alpha, low-affinity (Granulocyte-Macrophage); CSF2RAX; Granulocyte-Macrophage
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P73083
Purity:  ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: CSF2RA; GMCSFR-Alpha; Prev. CSF2R; CDw116; AlphaGMR; CSF2RY; CD116; Granulocyte-Macrophage Colony-Stimulating Factor Receptor Alpha Chain; Colony Stimulating Factor 2 Receptor, Alpha, low-affinity (Granulocyte-Macrophage); CSF2RAX; Granulocyte-Macrophage
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P73318
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: NGFR; low affinity Neurotrophin Receptor P75NTR; Nerve Growth Factor Receptor; TNFR Superfamily, Member 16; TNFRSF16; NGF Receptor; P75NTR; Gp80-LNGFR; CD271; P75 ICD; Tumor Necrosis Factor Receptor Superfamily Member 16; Nerve Growth Factor Receptor (TNF
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P74699
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: NGFR; low affinity Neurotrophin Receptor P75NTR; Nerve Growth Factor Receptor; TNFR Superfamily, Member 16; TNFRSF16; NGF Receptor; P75NTR; Gp80-LNGFR; CD271; P75 ICD; Tumor Necrosis Factor Receptor Superfamily Member 16; Nerve Growth Factor Receptor (TNF
Species:  
Rabbit
Source:  
HEK293
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Cat. No.: HY-P74700
Purity:  ≥ 85%, as determined by reducing SDS-PAGE.
Synonyms: NGFR; low affinity Neurotrophin Receptor P75NTR; Nerve Growth Factor Receptor; TNFR Superfamily, Member 16; TNFRSF16; NGF Receptor; P75NTR; Gp80-LNGFR; CD271; P75 ICD; Tumor Necrosis Factor Receptor Superfamily Member 16; Nerve Growth Factor Receptor (TNF
Species:  
Rabbit
Source:  
HEK293
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Cat. No.: HY-P77100
Purity:  ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: NGFR; low affinity Neurotrophin Receptor P75NTR; Nerve Growth Factor Receptor; TNFR Superfamily, Member 16; TNFRSF16; NGF Receptor; P75NTR; Gp80-LNGFR; CD271; P75 ICD; Tumor Necrosis Factor Receptor Superfamily Member 16; Nerve Growth Factor Receptor (TNF
Species:  
Mouse
Source:  
HEK293
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Cat. No.: HY-P77101
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: NGFR; low affinity Neurotrophin Receptor P75NTR; Nerve Growth Factor Receptor; TNFR Superfamily, Member 16; TNFRSF16; NGF Receptor; P75NTR; Gp80-LNGFR; CD271; P75 ICD; Tumor Necrosis Factor Receptor Superfamily Member 16; Nerve Growth Factor Receptor (TNF
Species:  
Mouse
Source:  
HEK293
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Cat. No.: HY-P77909
Purity:  ≥ 95%, as determined by Bis-Tris PAGE.
Synonyms: CSF2RA; GMCSFR-Alpha; Prev. CSF2R; CDw116; AlphaGMR; CSF2RY; CD116; Granulocyte-Macrophage Colony-Stimulating Factor Receptor Alpha Chain; Colony Stimulating Factor 2 Receptor, Alpha, low-affinity (Granulocyte-Macrophage); CSF2RAX; Granulocyte-Macrophage
Species:  
Mouse
Source:  
HEK293
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Cat. No.: HY-P700730
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: CSF2RA; GMCSFR-Alpha; Prev. CSF2R; CDw116; AlphaGMR; CSF2RY; CD116; Granulocyte-Macrophage Colony-Stimulating Factor Receptor Alpha Chain; Colony Stimulating Factor 2 Receptor, Alpha, low-affinity (Granulocyte-Macrophage); CSF2RAX; Granulocyte-Macrophage
Species:  
Cynomolgus
Source:  
HEK293
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Cat. No.: HY-135276A
Target:  

MicroRNA Apoptosis

Research Areas:  

Cancer

Targaprimir-96 TFA is a potent inhibitor of microRNA-96 (miR-96) processing. Targaprimir-96 TFA selectively modulates miR-96 production in cancer cells and triggers apoptosis. Targaprimir-96 TFA binds primary miR-96 (pri-miR-96) with low nanomolar affinity. Targaprimir-96 TFA directly engages pri-miR-96 in breast cancer cells and is ineffective on healthy breast cells .
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Cat. No.: HY-D1755
CAS No.: 348079-13-0
Fluo-3FF AM is a low affinity (Kd = 42 μM) fluorescent Ca 2+ sensitive indicator (Abs/Em = 462 nm/526 nm). Fluo-3FF AM is Mg 2+ insensitive and relatively photostable. Fluo-3FF AM is an analog of Fluo-3FF AM. Fluo-3FF AM is essentially non-fluorescent, but exhibits a strong fluorescence enhancement upon entry into cells and binding to calcium.
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Cat. No.: HY-P990827

Target:  

TROP2

Research Areas:  

Cancer

Anti-TROP-2 Antibody (Pr1E11) is a kind of mouse IgG1 κ chimeric antibody inhibitor, targeting to human TROP-2. Anti-TROP-2 Antibody (Pr1E11) specifically binds to TROP-2 with high affinity and shows low internalization activitv. Anti-TROP-2 Antibody (Pr1E11) can be used for the research of cancer, such as epithelial cancer and primary pancreatic cancer .
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Cat. No.: HY-P7269
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: PPBP; Macrophage-Derived Growth Factor; Prev. THBGB1; C-X-C Motif Chemokine 7; SCYB7; Beta-Thromboglobulin; CTAP3; NAP-2-L1; CXCL7; Small Inducible Cytokine Subfamily B, Member 7; MDGF; Neutrophil-Activating Peptide-2; LDGF; low-affinity Platelet Factor I
Species:  
Rat
Source:  
E. coli
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Cat. No.: HY-P78110
Purity:  ≥ 95%, as determined by Bis-Tris PAGE.
Synonyms: CSF2RA; GMCSFR-Alpha; Prev. CSF2R; CDw116; AlphaGMR; CSF2RY; CD116; Granulocyte-Macrophage Colony-Stimulating Factor Receptor Alpha Chain; Colony Stimulating Factor 2 Receptor, Alpha, low-affinity (Granulocyte-Macrophage); CSF2RAX; Granulocyte-Macrophage
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P87429A
Synonyms: CD16b, CD16B, FCG3, FCGR3, IGFR3, FCGR3B, low affinity immunoglobulin gamma Fc region receptor III-B, Fc-gamma RIII-beta, FcR-10, IgG Fc receptor III-1, CD16-I, Fc-gamma RIII, Fc-gamma RIIIb, FcRIII, FcRIIIb

Host:  

Mouse

Application:  

FC, ELISA

Reactivity:  

Human

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