2. GPCR/G Protein
  3. Vasopressin Receptor
  4. SKF 100398

SKF 100398  (Synonyms: d(CH2)5Tyr(Et)VAVP)

Cat. No.: HY-P3066 Purity: 99.25%
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SKF 100398 (d(CH2)5Tyr(Et)VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP.

For research use only. We do not sell to patients.

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SKF 100398 Chemical Structure

SKF 100398 Chemical Structure

CAS No. : 77453-01-1

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Description

SKF 100398 (d(CH2)5Tyr(Et)VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP[1].

In Vivo

SKF 100398 is a specific antagonist of the hydrosmotic effect of exogenous and endogenous AVP[1].
SKF 100398 (8 μg/kg; i.v.) abolishes the antidiuretic effect of AVP[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male Sprague-Dawley rats (250-300 g)[1]
Dosage: 8 μg/kg
Administration: Intravenous injection
Result: Completely blocked the antidiuretic effect of exogenous AVP (4 ng/kg body wt i.v.).
Molecular Weight

1136.39

Formula

C53H77N13O11S2
CAS No.
Appearance

Solid

Color

White to off-white

Sequence

{(1-Mercaptocyclohexyl)acetyl}-{Tyr(O-Ethyl)}-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge: 1-Cys6)
Sequence Shortening

{(1-Mercaptocyclohexyl)acetyl}-{Tyr(O-Ethyl)}-YFVNCPRG-NH2 (Disulfide bridge: 1-Cys6)
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Purity & Documentation

Purity: 99.25%

COA (262 KB) RP-HPLC (361 KB) LCMS (116 KB)

Handling Instructions (2659 KB)
References
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SKF 100398 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SKF 10039877453-01-1d(CH2)5Tyr(Et)VAVPSKF100398SKF-100398Vasopressin ReceptorargininevasopressinanalogueantidiureticactionInhibitorinhibitorinhibit

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